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peptide

Semaglutide

strongFDA-Approved· RxInjectionOral

Active ingredient in Ozempic/Wegovy. Mimics GLP-1 to signal fullness and slow gastric emptying. STEP trials showed 14.9% weight loss at 68 weeks.


Key facts
Classification
Semaglutide is a GLP-1 receptor agonist with Aib at position 8 for DPP-4 resistance and a C-18 fatty diacid chain enabling albumin binding (~7-day half-life).
Primary benefits
Fat Loss (10/10) · Longevity (5/10) · Gut Health (4/10)
Administration
Injection, Oral
Doses studied
Start at 0.25 mg per week subq and gradually increase to 1-2.4 mg per week over several months. An FDA-approved oral formulation (Rybelsus) is also available at 3-14 mg daily. Meant for long-term use.
Evidence strength
Strong — 21 peer-reviewed studies
Stacks well with
5-Amino-1MQ, BPC-157, MOTS-c
Legal status
FDA-Approved · prescription required · WADA prohibited
Quick stats
Type
Peptide
Administration
Injection, Oral
Studies referenced
21
Stacks with
3 peptides
Regulatory
FDA-Approved
Scientific overview

Semaglutide is a GLP-1 receptor agonist with Aib at position 8 for DPP-4 resistance and a C-18 fatty diacid chain enabling albumin binding (~7-day half-life). Enhances glucose-dependent insulin secretion, suppresses glucagon, delays gastric emptying, and reduces appetite via hypothalamic GLP-1 receptors. STEP 1 showed 14.9% weight reduction at 68 weeks.

Goal coverage · Semaglutide
🔥 Fat Loss10/10
Longevity5/10
🫃 Gut Health4/10
🧊 Inflammation3/10
FIG.1  Modeled goal coverage from reviewed studies. Score out of 10.
Medical oversight requiredNot safe during pregnancy· 6 contraindications
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