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capsule

Tesofensine

emergingPhase 2/3 Clinical TrialsOral

Originally for Parkinson's/Alzheimer's, found to cause major weight loss. Boosts serotonin, dopamine, and norepinephrine simultaneously, crushing appetite and revving metabolism.


Key facts
Classification
Tesofensine is a triple monoamine reuptake inhibitor (5-HT, NE, DA).
Primary benefits
Fat Loss (7/10) · Brain & Cognition (4/10) · Mood & Anxiety (3/10)
Administration
Oral
Doses studied
0.25-0.5 mg by mouth daily. Start at the lower dose. Cycle for 12-24 weeks.
Evidence strength
Emerging — 20 peer-reviewed studies
Stacks well with
Semaglutide, 5-Amino-1MQ
Legal status
Phase 2/3 Clinical Trials · not prescribable in US
Quick stats
Type
Capsule
Administration
Oral
Studies referenced
20
Stacks with
2 peptides
Regulatory
Phase 2/3 Clinical Trials
Scientific overview

Tesofensine is a triple monoamine reuptake inhibitor (5-HT, NE, DA). Phase 2 obesity trials showed 4.5-10.6% weight loss over 24 weeks via central appetite suppression and thermogenesis. Requires cardiovascular monitoring due to modest HR and BP increases.

Goal coverage · Tesofensine
🔥 Fat Loss7/10
🧠 Brain & Cognition4/10
😌 Mood & Anxiety3/10
FIG.1  Modeled goal coverage from reviewed studies. Score out of 10.
Medical oversight requiredNot safe during pregnancy· 7 contraindications
From our network:Cornerstone Peptide